Mecillinam


Mecillinam er et β-lactamantibiotikum i penicillingruppen med virkning på Gram-negative bakterier. Mecillinam har meget lav oral biotilgængelighed og derfor blev der udviklet et mere oralt aktivt prodrug, pivmecillinam. Pivmecillinam er pivaloyloxymethyl esteren til mecillinam og omdannes til mecillinam i organismen.
Mecillinam må administreres parenteralt og findes derfor kun som injektionsvæske, mens pivmecillinam findes som tabletter.
Anvendelse
Indikationer for behandling med mecillinam/pivmecillinam omfatter:
Præparater
Mecillinam er markedsført i Danmark under navnet Selexid®.
Pivmecillinam er markedsført i Danmark under navnene Selexid® og Penomax®.
Eksterne henvisninger
- Læs uddybende information om medicin, der indeholder Mecillinam på medicin.dk
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